SCHEMBL21947547

SCHEMBL21947547

COc1ccc(S(=O)(=O)NC2CCOC2)cc1C(=O)Nc1ccc(F)c(F)c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 11/20 0.60
HTR2B P41595 1/20 0.59
TP53 P04637 12/20 0.54
LMNA P02545 8/20 0.54
POLB P06746 1/20 0.48
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21569279 1.00 MAPT (0.60) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545409 0.93 HTR2B (0.69) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545406 0.93 HTR2B (0.69) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545347 0.92 HTR2B (0.54) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545349 0.92 HTR2B (0.54) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545661 0.92 HTR2B (0.56) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545662 0.92 HTR2B (0.56) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21947478 0.92 MAPT (0.53) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21569514 0.92 MAPT (0.53) MAPTHTR2BTP53LMNAPOLB
SCHEMBL21545343 0.91 HTR2B (0.56) MAPTHTR2BTP53LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10654837-B2 Sulphamoylaryl derivatives and use thereof as medicaments for the treatment of liver fibrosis JANSSEN PHARMACEUTICA NV (BE) 2020-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10654837-B2 Sulphamoylaryl derivatives and use thereof as medicaments for the treatment of liver fibrosis HTR2B, HTR3B, HTR1A MAPT 4615/4885HTR2B 1/4885TP53 3645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.