SCHEMBL21964516

SCHEMBL21964516

CC/C=C/N(C(=O)OC(C)(C)C)c1cccc(N)c1C

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.34
KCNH2 Q12809 1/20 0.34
CHEK1 O14757 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
PIK3CA P42336 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
GRM6 O15303 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20045665 0.77 CYP3A4 (0.39) ESR1KCNH2ALDH1A1HSD17B10CYP3A4
SCHEMBL30961659 0.77 CYP3A4 (0.39) ESR1KCNH2ALDH1A1HSD17B10CYP3A4
SCHEMBL28317708 0.72 ESR1 (0.34) ESR1KCNH2ALDH1A1CYP3A4TSHR
SCHEMBL6677666 0.70 ESR1 (0.42) ESR1KCNH2ALDH1A1HSD17B10CYP3A4
SCHEMBL5929895 0.69 ESR1 (0.40) ESR1KCNH2ALDH1A1HSD17B10CYP3A4
SCHEMBL6681404 0.69 ESR1 (0.41) ESR1KCNH2ALDH1A1HSD17B10CYP3A4
SCHEMBL16113033 0.68 ALDH1A1 (0.38) ALDH1A1HSD17B10CYP3A4TSHR
SCHEMBL1068685 0.67 ESR1 (0.42) ESR1KCNH2ALDH1A1HSD17B10CYP3A4
SCHEMBL29223984 0.67 GRM6 (0.38) ALDH1A1HSD17B10TSHRGRM6
SCHEMBL30864316 0.67 GRM6 (0.38) ALDH1A1HSD17B10TSHRGRM6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3643703-A1 EP300/CREBBP INHIBITOR Daiichi Sankyo Co., Ltd. (JP) 2020-04-29 EP disclosed