SCHEMBL21970124

SCHEMBL21970124

O=C1CC2CCc3cc(NCCO)ccc3C2=NN1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.48
KCNH2 Q12809 1/20 0.48
PDE3A Q14432 9/20 0.42
PDE3B Q13370 8/20 0.42
GALR3 O60755 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
GPR119 Q8TDV5 3/20 0.35
ABL1 P00519 1/20 0.34
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10900264 0.87 HRH3 (0.49) HRH3KCNH2PDE3APDE3BITGB3
SCHEMBL10753732 0.83 HRH3 (0.46) HRH3KCNH2PDE3APDE3BMAPT
SCHEMBL10341508 0.81 PDE3B (0.53) HRH3KCNH2PDE3APDE3BMAPT
SCHEMBL10341540 0.81 HRH3 (0.50) HRH3KCNH2PDE3APDE3BITGB3
SCHEMBL10740298 0.76 PDE3A (0.50) HRH3KCNH2PDE3APDE3BGALR3
SCHEMBL9602068 0.76 HRH3 (0.57) HRH3KCNH2PDE3APDE3BGALR3
SCHEMBL8305150 0.76 HRH3 (0.54) HRH3KCNH2PDE3APDE3BGPR119
SCHEMBL10753296 0.76 HRH3 (0.54) HRH3KCNH2PDE3APDE3B
Hydrochloric Acid SCHEMBL11092318 0.76 PDE3B (0.49) HRH3KCNH2PDE3APDE3BGALR3
Hydrochloric Acid SCHEMBL7314082 0.75 HRH3 (0.56) HRH3KCNH2PDE3APDE3BGALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970145-B1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CANCER BROAD INST INC (US) 2020-05-06 EP disclosed