SCHEMBL21971012

SCHEMBL21971012

CN1C(=O)c2ccccc2-c2cc(Cl)ccc2C12CC2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 2/20 0.42
CCR5 P51681 1/20 0.41
DRD2 P14416 3/20 0.40
DRD4 P21917 3/20 0.40
PDK2 Q15119 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PGR P06401 4/20 0.37
UTS2R Q9UKP6 1/20 0.36
AKR1B1 P15121 1/20 0.36
MDM2 Q00987 1/20 0.36
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21903270 0.84 NPC1 (0.40) S100A4CYP11B1CYP11B2MEN1KMT2A
SCHEMBL21903238 0.82 CYP11B2 (0.42) S100A4DRD2DRD4CYP11B1CYP11B2
SCHEMBL29986526 0.80 CYP11B2 (0.39) CCR5CYP11B1CYP11B2
SCHEMBL21970098 0.80 CYP11B2 (0.39) CCR5CYP11B1CYP11B2
SCHEMBL30372076 0.80 HRH3 (0.51) CCR5HRH3MEN1KMT2APGR
SCHEMBL21903272 0.75 MAP3K5 (0.39) HRH3
SCHEMBL22898412 0.74 NR1H2 (0.40) HRH3MEN1KMT2A
SCHEMBL21903240 0.74 MDM2 (0.36) CYP11B1CYP11B2AKR1B1MDM2
Hydrochloric Acid SCHEMBL29985745 0.74 MAP3K5 (0.39) HRH3
SCHEMBL30564277 0.73 HRH3 (0.52) CCR5HRH3MEN1KMT2APGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200140438-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AS ALLOSTERIC MODULATORS OF GROUP II METABOTROPIC GLUTAMATE RECEPTORS DOMAIN THERAPEUTICS (FR) 2020-05-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200140438-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AS ALLOSTERIC MODULATORS OF GROUP II METABOTROPIC GLUTAMATE RECEPTORS GRM3, GRM1, GRM2 S100A4 2264/4885CCR5 1987/4885DRD2 565/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.