SCHEMBL21974541

SCHEMBL21974541

CNc1ccc(-c2ccc(N)cc2COC(=O)/C=C/c2ccc(OC(=O)c3ccc(OCCCC(F)(F)F)cc3)cc2)c(COC(=O)/C=C/c2ccc(OC(=O)c3ccc(OCCCC(F)(F)F)cc3)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
APP P05067 10/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679372 0.93 ABCG2 (0.40) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL30086264 0.93 ABCG2 (0.40) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL18112629 0.93 ABCG2 (0.40) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL679305 0.86 MAPT (0.39) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL14019209 0.85 KMT2A (0.43) ABCG2KDM4EMAPTCA12CA1
SCHEMBL18993099 0.85 ABCG2 (0.35) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL3634719 0.85 ABCG2 (0.39) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL13829579 0.85 ABCG2 (0.39) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL2136229 0.85 ABCG2 (0.39) SAE1UBA2ABCG2KDM4EMAPT
SCHEMBL15771844 0.85 ABCG2 (0.34) ABCG2KDM4EMAPTCYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107978-B1 LIQUID CRYSTAL ALIGNMENT COMPOSITION, LIQUID CRYSTAL ALIGNMENT FILM AND LIQUID CRYSTAL DISPLAY ELEMENT ROLIC TECH AG (CH) 2020-05-06 EP disclosed