SCHEMBL21976231

SCHEMBL21976231

O=C(NO)c1ccc2c(c1)NC(c1cccc(-c3cccc(Cl)c3)c1)N2

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 6/20 0.47
HDAC8 Q9BY41 7/20 0.45
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MCL1 Q07820 1/20 0.42
HDAC1 Q13547 7/20 0.42
PLAU P00749 1/20 0.41
KAT6A Q92794 1/20 0.38
SMPD1 P17405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21976203 0.93 GAA (0.49) HDAC6HDAC8GAAMAPTMEN1
SCHEMBL21976963 0.92 HDAC6 (0.49) HDAC6HDAC8HDAC1PLAUSMPD1
SCHEMBL21976967 0.81 HDAC6 (0.47) HDAC6HDAC8MAPTHDAC1KAT6A
SCHEMBL21976470 0.80 HDAC6 (0.55) HDAC6HDAC8MEN1KMT2AHDAC1
SCHEMBL21976943 0.78 HDAC8 (0.52) HDAC6HDAC8MAPTHDAC1
SCHEMBL5943946 0.74 HDAC6 (0.61) HDAC6HDAC8MEN1KMT2AHDAC1
SCHEMBL21976479 0.74 HDAC6 (0.50) HDAC6HDAC8MAPTHDAC1SMPD1
SCHEMBL21976251 0.72 HDAC6 (0.52) HDAC6HDAC8HDAC1PLAUSMPD1
SCHEMBL21976950 0.71 HDAC1 (0.47) HDAC6HDAC8GAAHDAC1
SCHEMBL21976968 0.71 HDAC6 (0.50) HDAC6HDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed