SCHEMBL21976963

SCHEMBL21976963

O=C(NO)c1ccc2c(c1)NC(c1ccc(-c3cccc(Cl)c3)cc1)N2

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.49
HDAC8 Q9BY41 7/20 0.47
PLAU P00749 1/20 0.46
HDAC1 Q13547 3/20 0.42
GRM5 P41594 1/20 0.41
PARP1 P09874 1/20 0.41
SMPD1 P17405 1/20 0.39
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21976231 0.92 HDAC6 (0.47) HDAC6HDAC8PLAUHDAC1SMPD1
SCHEMBL21976203 0.87 GAA (0.49) HDAC6HDAC8HDAC1
SCHEMBL21976251 0.81 HDAC6 (0.52) HDAC6HDAC8PLAUHDAC1PARP1
SCHEMBL5943946 0.79 HDAC6 (0.61) HDAC6HDAC8PLAUHDAC1GRM5
SCHEMBL21975936 0.79 MEN1 (0.42) HDAC6HDAC8HDAC1MMP2MMP9
SCHEMBL21976309 0.77 HDAC6 (0.41) HDAC6HDAC8HDAC1
SCHEMBL21976503 0.74 MEN1 (0.45) HDAC6HDAC8HDAC1
SCHEMBL21976470 0.74 HDAC6 (0.55) HDAC6HDAC8HDAC1
SCHEMBL21976943 0.72 HDAC8 (0.52) HDAC6HDAC8HDAC1
SCHEMBL6674303 0.72 KDM4E (0.62) HDAC6HDAC8HDAC1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294715-B1 BENZIMIDAZOLE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN HISTONE DEACETYLASE ACTIVITY KANCERA AB (SE) 2020-05-06 EP disclosed