SCHEMBL2197752

SCHEMBL2197752

CS(=O)(=O)c1ccc(C(Oc2ccc(F)cc2F)c2cc3cccnc3[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GCK P35557 8/20 0.40
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
BRD4 O60885 4/20 0.38
TRPA1 O75762 1/20 0.36
MAPT P10636 1/20 0.36
GPR6 P46095 1/20 0.35
EPHX2 P34913 1/20 0.35
NR3C1 P04150 1/20 0.35
NR3C2 P08235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12490508 0.84 BRD4 (0.40) GCKPTGS2PTGS1BRD4MAPT
SCHEMBL12490119 0.80 GCK (0.46) GCKPTGS2PTGS1
SCHEMBL2195791 0.76 GCK (0.44) GCK
SCHEMBL2196134 0.74 GCK (0.47) GCK
SCHEMBL12489676 0.72 GPR6 (0.39) GCKPTGS2PTGS1BRD4GPR6
SCHEMBL1960655 0.70 GCK (0.52) GCK
SCHEMBL1959200 0.69 GCK (0.51) GCK
SCHEMBL2179681 0.69 GCK (0.48) GCKBRD4
SCHEMBL1962013 0.67 GCK (0.75) GCK
SCHEMBL2195649 0.67 GCK (0.45) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO disclosed