SCHEMBL21985368

SCHEMBL21985368

CNc1ncc(C)nc1N

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.34
PDPK1 O15530 1/20 0.33
MAPKAPK2 P49137 1/20 0.32
NOS3 P29474 2/20 0.31
NOS2 P35228 2/20 0.31
UHRF1 Q96T88 1/20 0.31
NOS1 P29475 1/20 0.31
MAP4K4 O95819 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ADORA2A P29274 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
NUDT1 P36639 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25763275 0.83 KDM4E (0.34) GRM5MAPKAPK2NOS3NOS2UHRF1
SCHEMBL18824620 0.78 ADORA2A (0.37) GRM5PDPK1MAP4K4ADORA2A
SCHEMBL31362142 0.78 ADORA2A (0.37) GRM5PDPK1MAP4K4ADORA2A
SCHEMBL17084504 0.77 JAK3 (0.35) PDPK1NOS3NOS2CYP1A2CYP3A4
SCHEMBL27180300 0.77 MAPKAPK2 (0.41) GRM5MAPKAPK2
SCHEMBL16346270 0.77 ADORA2A (0.33) PDPK1MAP4K4ADORA2A
SCHEMBL24457887 0.74 NOS3 (0.30) NOS3NOS2CYP1A2CYP3A4CYP2D6
SCHEMBL12648083 0.74
SCHEMBL30716708 0.74
SCHEMBL9926609 0.73 CYP3A4 (0.33) PDPK1NOS3NOS2KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778599-A2 PESTICIDALLY ACTIVE BI- OR TRICYCLIC HETEROCYCLES WITH SULFUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2021-02-17 EP disclosed
EP-3778598-A2 PESTICIDALLY ACTIVE BI- OR TRICYCLIC HETEROCYCLES WITH SULFUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2021-02-17 EP disclosed
EP-3016949-B1 PESTICIDALLY ACTIVE BI- OR TRICYCLIC HETEROCYCLES WITH SULFUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2020-05-13 EP disclosed