SCHEMBL21987015

SCHEMBL21987015

Oc1cccc2ccc(Cc3ccccc3)cc12

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.56
CYP1A2 P05177 2/20 0.50
CTDSP1 Q9GZU7 1/20 0.50
HNF4A P41235 1/20 0.49
OPRK1 P41145 1/20 0.47
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
BCL2 P10415 1/20 0.46
BCL2L1 Q07817 1/20 0.46
MPO P05164 1/20 0.44
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ACMSD Q8TDX5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922542 0.86 IDH1 (0.56) IDH1CYP1A2HNF4ABCL2BCL2L1
SCHEMBL24928859 0.84
SCHEMBL26003882 0.83
SCHEMBL27877433 0.81 ALDH1A1 (0.54) IDH1CYP1A2PRSS1PRSS2PRSS3
SCHEMBL16846166 0.79
SCHEMBL2056356 0.78 CYP1A2 (0.53) CYP1A2CTDSP1HSD17B10
SCHEMBL15345371 0.78 CTDSP1 (0.58) CYP1A2CTDSP1
SCHEMBL21585559 0.77 AKR1B1 (0.58) CYP1A2CTDSP1CYP2C19HSD17B10
SCHEMBL15345635 0.76 PRSS1 (0.44) IDH1CYP1A2PRSS1PRSS2PRSS3
SCHEMBL27919165 0.76 TRPV1 (0.42) IDH1PRSS1PRSS2PRSS3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3659593-A1 TRMT2A INHIBITORS FOR USE IN THE TREATMENT OF POLYGLUTAMINE DISEASES Forschungszentrum Jülich GmbH/ Abteilung RP-PT (DE) 2020-06-03 EP disclosed