SCHEMBL21992124

SCHEMBL21992124

Cc1cc(F)cc(N(C)C(=O)[C@@H](C)Cc2cc(F)cc(F)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.35
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
MAOB P27338 1/20 0.34
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
BACE1 P56817 4/20 0.32
BACE2 Q9Y5Z0 3/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
GRM5 P41594 1/20 0.31
SLC6A3 Q01959 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18179962 0.85 SLC7A5 (0.36) NR3C1PGRNR3C2MAOBNOS3
SCHEMBL19999803 0.80 HPGD (0.36) HPGDMAOB
SCHEMBL21993361 0.80 HPGD (0.36) HPGDMAOBKMT2AMEN1LMNA
SCHEMBL21992337 0.80 MAOB (0.39) HPGDMAOBBACE1KMT2AMEN1
SCHEMBL19962120 0.80 HPGD (0.38) HPGDMAOBKMT2AMEN1SLC6A3
SCHEMBL21993366 0.78 MAOB (0.40) HPGDMAOBKMT2AMEN1LMNA
SCHEMBL19999802 0.78 S1PR1 (0.41) HPGDMAOBKMT2AMEN1
SCHEMBL21992634 0.78 SMN1; SMN2 (0.39) HPGDMAOBSLC6A3
SCHEMBL21992128 0.77 MAOB (0.37) HPGDMAOBKMT2ALMNA
SCHEMBL19999809 0.77 MAOB (0.38) HPGDMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286166-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2020-05-13 EP disclosed