SCHEMBL21992128

SCHEMBL21992128

CCCc1ccc(N(C)C(=O)[C@@H](C)Cc2cc(F)cc(F)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
HPGD P15428 1/20 0.36
PER2 O15055 1/20 0.36
CRY1 Q16526 1/20 0.36
CRY2 Q49AN0 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GPR88 Q9GZN0 1/20 0.35
MLYCD O95822 1/20 0.35
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21992337 0.90 MAOB (0.39) MAOBHPGDPER2CRY1CRY2
SCHEMBL19962121 0.86 CIT (0.38) MAOBESR1ESR2PER2CRY1
SCHEMBL21993366 0.86 MAOB (0.40) MAOBHPGDCRY1CRY2ALDH1A1
SCHEMBL19999809 0.82 MAOB (0.38) MAOBHPGDGPR88MLYCD
SCHEMBL19962120 0.82 HPGD (0.38) MAOBHPGDKMT2ALMNAGPR88
SCHEMBL19999803 0.80 HPGD (0.36) MAOBHPGDGPR88MLYCD
SCHEMBL21993361 0.80 HPGD (0.36) MAOBHPGDALDH1A1KMT2ALMNA
SCHEMBL21992634 0.78 SMN1; SMN2 (0.39) MAOBHPGDALDH1A1NPC1RAB9A
SCHEMBL19999802 0.78 S1PR1 (0.41) MAOBHPGDALDH1A1KMT2ATDP1
SCHEMBL21992124 0.77 HPGD (0.35) MAOBHPGDKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286166-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2020-05-13 EP disclosed