SCHEMBL2199213

SCHEMBL2199213

COC(=O)c1ccc(OC)c(C(=O)c2ccc(Nc3ccc(F)cc3F)cc2Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.54
EGFR P00533 1/20 0.54
MET P08581 1/20 0.54
MAPK13 O15264 2/20 0.53
MAPK12 P53778 2/20 0.53
MAPK11 Q15759 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.48
RAB9A P51151 2/20 0.48
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
PYGL P06737 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2203119 0.92 MAPK14 (0.54) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2199146 0.92 MAPK14 (0.54) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2201621 0.91 MAPK14 (0.53) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2199428 0.89 MAPK14 (0.60) MAPK14MAPK13MAPK12MAPK11SMN1; SMN2
SCHEMBL2198797 0.89 MAPK14 (0.62) MAPK14MAPK13MAPK12MAPK11SMN1; SMN2
SCHEMBL2200130 0.89 MAPK14 (0.52) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2852568 0.87 MAPK14 (0.53) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2198633 0.86 MAPK14 (0.51) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2198978 0.86 MAPK14 (0.51) MAPK14EGFRMETMAPK13MAPK12
SCHEMBL2196670 0.86 MAPK14 (0.51) MAPK14EGFRMETMAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658263-B9 NOVEL AMINOBENZOPHENONE COMPOUNDS LEO PHARMA AS (DK) 2011-11-09 EP disclosed
US-7977387-B2 Aminobenzophenone compounds LEO PHARMA A/S (DK) 2011-07-12 US disclosed
EP-1658263-B1 NOVEL AMINOBENZOPHENONE COMPOUNDS LEO PHARMA AS (DK) 2010-06-02 EP disclosed
US-20060166990-A1 Novel aminobenzophenone compounds LEO PHARMA A/S (DK) 2006-07-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060166990-A1 Novel aminobenzophenone compounds NFKBIA, UACA, ALDH7A1 MAPK14 697/4885EGFR 591/4885MET 1973/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.