SCHEMBL21996491

SCHEMBL21996491

CC(C)(C)OC(=O)N1C[C@@H](OCc2cc(F)c(F)c(F)c2)CC12C=C2

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.35
SIGMAR1 Q99720 3/20 0.35
TMEM97 Q5BJF2 2/20 0.35
BACE1 P56817 2/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
USP30 Q70CQ3 1/20 0.33
AOC3 Q16853 1/20 0.33
DPP4 P27487 1/20 0.32
MAOB P27338 1/20 0.32
SCN9A Q15858 2/20 0.32
GPR119 Q8TDV5 4/20 0.32
TACR1 P25103 1/20 0.32
PAK1 Q13153 1/20 0.31
DRD3 P35462 2/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22047547 1.00 DRD4 (0.35) DRD4SIGMAR1TMEM97BACE1BACE2
SCHEMBL22047120 0.87 BACE1 (0.34) DRD4SIGMAR1TMEM97BACE1BACE2
SCHEMBL21996612 0.86 USP30 (0.34) DRD4SIGMAR1TMEM97BACE1BACE2
SCHEMBL24622151 0.86 BACE1 (0.39) BACE1BACE2DDB1CRBN
SCHEMBL21996313 0.86 BACE1 (0.39) BACE1BACE2DDB1CRBN
SCHEMBL21996540 0.84 USP30 (0.33) DRD4SIGMAR1TMEM97BACE1BACE2
SCHEMBL21996508 0.83 ABCB1 (0.41) BACE1BACE2GPR119DDB1CRBN
SCHEMBL24622152 0.83 ABCB1 (0.41) BACE1BACE2GPR119DDB1CRBN
SCHEMBL24622085 0.81 BACE1 (0.36) BACE1BACE2DDB1CRBN
SCHEMBL22323665 0.76 BACE1 (0.36) DRD4SIGMAR1TMEM97BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020113077-A9 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-08-13 WO disclosed
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed