SCHEMBL21996510

SCHEMBL21996510

C=C1C[C@H](OCc2cc(F)c(F)c(F)c2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.36
BACE2 Q9Y5Z0 1/20 0.35
USP30 Q70CQ3 2/20 0.34
DPP4 P27487 1/20 0.33
MAOB P27338 1/20 0.33
GPR119 Q8TDV5 3/20 0.32
DRD4 P21917 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
TACR1 P25103 3/20 0.32
SCN9A Q15858 1/20 0.31
RIPK1 Q13546 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22323665 1.00 BACE1 (0.36) BACE1BACE2USP30DPP4MAOB
SCHEMBL22047155 0.86 BACE1 (0.43) BACE1BACE2TACR1LIPGHDAC1
SCHEMBL21996478 0.86 BACE1 (0.43) BACE1BACE2TACR1LIPGHDAC1
SCHEMBL22324617 0.82 ABCB1 (0.42) BACE1BACE2GPR119
SCHEMBL21996514 0.82 ABCB1 (0.42) BACE1BACE2GPR119
SCHEMBL21996445 0.76 ABCB1 (0.43) BACE1BACE2DPP4MAOBGPR119
SCHEMBL22047120 0.76 BACE1 (0.34) BACE1BACE2USP30DPP4MAOB
SCHEMBL22047547 0.76 DRD4 (0.35) BACE1BACE2USP30DPP4MAOB
SCHEMBL21996491 0.76 DRD4 (0.35) BACE1BACE2USP30DPP4MAOB
SCHEMBL21996612 0.75 USP30 (0.34) BACE1BACE2USP30DPP4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed