SCHEMBL21996539

SCHEMBL21996539

COC(=O)C1CC(OCc2ccc(F)cc2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.44
ABCB1 P08183 1/20 0.43
BACE1 P56817 2/20 0.42
BACE2 Q9Y5Z0 1/20 0.42
GPR119 Q8TDV5 2/20 0.40
MCL1 Q07820 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
AGTR2 P50052 1/20 0.39
KLK7 P49862 1/20 0.38
PTPN1 P18031 1/20 0.38
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
CCR3 P51677 1/20 0.38
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
MMP1 P03956 1/20 0.37
ADAM17 P78536 1/20 0.37
UCHL1 P09936 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3857592 0.89 P2RX3 (0.48) P2RX3ABCB1GPR119MCL1MMP1
SCHEMBL3190398 0.89 P2RX3 (0.54) P2RX3ABCB1GPR119MCL1NR1H2
SCHEMBL8170628 0.89 P2RX3 (0.54) P2RX3ABCB1GPR119MCL1NR1H2
SCHEMBL27043958 0.89 P2RX3 (0.48) P2RX3ABCB1GPR119MCL1MMP1
SCHEMBL12028132 0.89 MCL1 (0.44) P2RX3ABCB1GPR119MCL1NR1H2
SCHEMBL475487 0.89 ABCB1 (0.52) P2RX3ABCB1MCL1NR1H2NR1H3
SCHEMBL3191348 0.89 ABCB1 (0.52) P2RX3ABCB1MCL1NR1H2NR1H3
SCHEMBL475486 0.89 ABCB1 (0.52) P2RX3ABCB1MCL1NR1H2NR1H3
SCHEMBL3854950 0.89 ABCB1 (0.52) P2RX3ABCB1MCL1NR1H2NR1H3
SCHEMBL18093988 0.89 ABCB1 (0.52) P2RX3ABCB1MCL1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020113077-A9 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-08-13 WO disclosed
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed
WO-2020113077-A1 COMPOSITIONS AND METHODS FOR MODULAR CONTROL OF BIOORTHOGONAL LIGATION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-06-04 WO disclosed