SCHEMBL2200303

SCHEMBL2200303

CC(=O)NC1CCN(C2CCN(C(=O)c3c(C)nn(-c4cccc(OC(F)(F)F)c4)c3C)C2)C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
SMPD3 Q9NY59 1/20 0.43
NPY5R Q15761 1/20 0.39
NOTUM Q6P988 1/20 0.38
SCN9A Q15858 3/20 0.38
ACACB O00763 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
RECQL P46063 1/20 0.37
PRKAA2 P54646 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PIM1 P11309 2/20 0.36
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2201420 0.96 KMT2A (0.47) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL2200867 0.96 KMT2A (0.47) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL2201606 0.96 KMT2A (0.47) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL2202314 0.89 KMT2A (0.47) KMT2ANPY5RNOTUMSCN9ASCN10A
SCHEMBL2202211 0.89 KMT2A (0.47) KMT2ANPY5RNOTUMSCN9ASCN10A
SCHEMBL2202124 0.88 SMPD3 (0.41) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL2201293 0.88 SMPD3 (0.41) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL2201296 0.88 SMPD3 (0.41) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL12429652 0.86 KMT2A (0.44) KMT2ASMPD3NPY5RNOTUMSCN9A
SCHEMBL2201084 0.84 KMT2A (0.49) KMT2ANPY5RNOTUMSCN9ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977358-B2 Pyrazol derivatives HOFFMANN-LA ROCHE INC. (US) 2011-07-12 US disclosed
US-20090029963-A1 PYRAZOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090029963-A1 PYRAZOL DERIVATIVES CCR1, CCR3, CCRL2 KMT2A 4057/4885SMPD3 3106/4885NPY5R 277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.