SCHEMBL22005109

SCHEMBL22005109

COC(=O)c1cc2c(cc1Cl)cc(-c1cncnc1)n2C(C)C

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACLY P53396 4/20 0.56
MAOA P21397 1/20 0.37
P2RX3 P56373 1/20 0.36
NR4A2 P43354 2/20 0.35
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ABL1 P00519 3/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22005117 0.87 ACLY (0.53) ACLYMAOAMAPTKMT2AKDM4E
SCHEMBL22005107 0.85 ACLY (0.59) ACLYMAOANR4A2MAPTNPSR1
SCHEMBL22004320 0.78 MAPT (0.41) ACLYMAOAP2RX3MAPTNPSR1
SCHEMBL22004214 0.72 ACLY (1.00) ACLY
SCHEMBL22004122 0.71 ACLY (0.46) ACLYMAPTHTR2AHTR2CKMT2A
SCHEMBL22005118 0.71 ACLY (0.55) ACLYMAOAKMT2A
SCHEMBL17185620 0.68 PDK2 (0.48) ACLYNR4A2MAPTABL1KDM4E
SCHEMBL8706096 0.68 ACLY (0.46) ACLYNR4A2MAPTNPSR1ABL1
SCHEMBL22005105 0.67 ACLY (0.46) ACLYMAPTABL1HTR2AHTR2C
SCHEMBL22005030 0.67 ACLY (0.40) ACLYMAPTKMT2AHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200157076-A1 ACLY INHIBITORS AND USES THEREOF NIMBUS DISCOVERY, INC. 2020-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200157076-A1 ACLY INHIBITORS AND USES THEREOF ACLY, ATP5ME, ATP5MG ACLY 1/4885MAOA 3294/4885P2RX3 1422/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.