SCHEMBL22010383

SCHEMBL22010383

CC/C=C\CCS(=N)(N)=O

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
CYP19A1 P11511 2/20 0.33
RXRA P19793 2/20 0.33
PPARG P37231 2/20 0.33
OXER1 Q8TDS5 2/20 0.33
FFAR1 O14842 1/20 0.33
MAPT P10636 1/20 0.33
PPARA Q07869 2/20 0.32
F7 P08709 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
F3 P13726 1/20 0.31
PTGS1 P23219 1/20 0.31
KMT2A Q03164 1/20 0.31
PPARD Q03181 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28134376 0.81 ALDH1A1 (0.35) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL8989609 0.75 ALDH1A1 (0.38) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL11301760 0.75 ALDH1A1 (0.38) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL10978361 0.71 EPHX2 (0.41) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL19526875 0.69
SCHEMBL20376216 0.68 ALDH1A1 (0.33) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL14617949 0.65 ALDH1A1 (0.41) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL2363271 0.64 ALDH1A1 (0.43) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL19751288 0.64 ALDH1A1 (0.43) ALDH1A1CYP19A1RXRAPPARGOXER1
SCHEMBL2363268 0.64 ALDH1A1 (0.43) ALDH1A1CYP19A1RXRAPPARGOXER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102100-A9 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-01-06 WO disclosed
WO-2020102100-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed