SCHEMBL22010469

SCHEMBL22010469

CC(C)(C)OC(=O)N1CC2C=C(c3ccc(Oc4ccncc4)cc3)CC2C1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 4/20 0.47
CCNT1 O60563 2/20 0.44
CDK9 P50750 2/20 0.44
GPR119 Q8TDV5 5/20 0.41
TNK2 Q07912 1/20 0.38
GRM1 Q13255 1/20 0.38
GRM2 Q14416 1/20 0.38
NR1H2 P55055 1/20 0.38
USP30 Q70CQ3 1/20 0.38
LIPE Q05469 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22010468 1.00 BTK (0.47) BTKCCNT1CDK9GPR119TNK2
SCHEMBL15803566 0.91 CCNT1 (0.47) CCNT1CDK9GPR119GRM1GRM2
SCHEMBL15803568 0.91 CCNT1 (0.47) CCNT1CDK9GPR119GRM1GRM2
SCHEMBL15803567 0.91 CCNT1 (0.47) CCNT1CDK9GPR119GRM1GRM2
SCHEMBL30161685 0.89 BTK (0.52) BTKCCNT1CDK9GPR119TNK2
SCHEMBL22010906 0.89 BTK (0.52) BTKCCNT1CDK9GPR119TNK2
SCHEMBL22010736 0.88 BTK (0.45) BTKCCNT1CDK9GPR119TNK2
SCHEMBL22010483 0.88 BTK (0.45) BTKCCNT1CDK9GPR119TNK2
SCHEMBL22010485 0.88 BTK (0.45) BTKCCNT1CDK9GPR119TNK2
SCHEMBL22010769 0.85 GPR119 (0.48) BTKCCNT1CDK9GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020099341-A1 ANTIBIOTIC COMPOUNDS, METHODS OF MANUFACTURING THE SAME, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND USES THEREOF DEBIOPHARM INTERNATIONAL S.A. (CH) 2020-05-22 WO disclosed