SCHEMBL22013250

SCHEMBL22013250

OCCNc1ccnc2ccc(N3CCCC3)nc12

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.45
CXCR4 P61073 1/20 0.44
SLC29A1 Q99808 3/20 0.44
SORD Q00796 1/20 0.41
GBA1 P04062 9/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23837044 0.80 MAP4K4 (0.50) MAP4K4CXCR4
SCHEMBL22014121 0.76 KIT (0.46)
SCHEMBL22013645 0.73 MAP4K4 (0.55) MAP4K4CXCR4SORD
SCHEMBL22013086 0.73 NTRK1 (0.51)
SCHEMBL29692877 0.73 NTRK1 (0.51)
SCHEMBL29692833 0.73 NTRK1 (0.51)
SCHEMBL22013243 0.72 MAPK8 (0.47) MAP4K4MKNK1MKNK2
SCHEMBL22013643 0.72 MAP4K4 (0.61) MAP4K4CXCR4
SCHEMBL23836983 0.72 MAP4K4 (0.54) MAP4K4GBA1
SCHEMBL22013226 0.72 MAP4K4 (0.54) MAP4K4CXCR4SORD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882247-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-09-22 EP disclosed
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed