SCHEMBL22013645

SCHEMBL22013645

c1cc(N2CCCC2)c2nc(N3CCCC3)ccc2n1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 10/20 0.55
PKM P14618 1/20 0.45
ALOX15 P16050 1/20 0.45
CASP1 P29466 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CHKA P35790 1/20 0.44
CXCR4 P61073 1/20 0.40
SORD Q00796 1/20 0.40
MAOB P27338 4/20 0.39
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23837016 0.84 PDE10A (0.45) MAP4K4PDE10A
SCHEMBL22013375 0.84 PDE10A (0.45) MAP4K4PDE10A
SCHEMBL22013226 0.82 MAP4K4 (0.54) MAP4K4PKMALOX15CASP1HSD17B10
SCHEMBL22013643 0.82 MAP4K4 (0.61) MAP4K4CXCR4
SCHEMBL23836983 0.82 MAP4K4 (0.54) MAP4K4HSD17B10
SCHEMBL23837030 0.78 MAP4K4 (0.50) MAP4K4
SCHEMBL23837044 0.78 MAP4K4 (0.50) MAP4K4CXCR4
SCHEMBL22013653 0.76 MAP4K4 (0.51) MAP4K4
SCHEMBL22014120 0.73 MAP4K4 (0.45) MAP4K4PKM
SCHEMBL22013250 0.73 MAP4K4 (0.45) MAP4K4CXCR4SORD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3882247-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR Shanghai Ennovabio Pharmaceuticals Co., Ltd. (CN) 2021-09-22 EP disclosed
WO-2020098723-A1 SIX-MEMBERED AND SIX-MEMBERED HETEROCYCLIC COMPOUND AND USES THEREOF SERVING AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed