SCHEMBL22013636

SCHEMBL22013636

CC(C)(C)[Si](C)(C)NS(=O)(=O)c1ccc(Br)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NMT1 P30419 1/20 0.52
PFKFB4 Q16877 1/20 0.44
AKR1B1 P15121 1/20 0.43
APLNR P35414 2/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
PPARG P37231 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.39
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
EIF2AK3 Q9NZJ5 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
RRM1 P23921 1/20 0.36
RRM2B Q7LG56 1/20 0.36
ALPL P05186 1/20 0.36
JAK1 P23458 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20680929 0.82 NMT1 (0.36) NMT1CHRM2CHRM1RRM1RRM2B
SCHEMBL14930239 0.78 NMT1 (0.54) NMT1PFKFB4AKR1B1CA1CA2
SCHEMBL2371748 0.77 NMT1 (0.56) NMT1PFKFB4AKR1B1CA1CA2
SCHEMBL21893271 0.76 PIK3CA (0.37) NMT1CA2TSHR
SCHEMBL25389850 0.76 SLC22A12 (0.35) NMT1ALPLKMT2A
SCHEMBL31347243 0.75 IDO1 (0.40) PPARGCYP3A4CYP2C9TSHRJAK1
SCHEMBL30562770 0.74 EDNRB (0.50) KMT2A
SCHEMBL25387423 0.74 EDNRB (0.50) KMT2A
SCHEMBL2371744 0.74 NMT1 (0.52) NMT1PFKFB4AKR1B1CA1CA2
SCHEMBL22012124 0.74 BRD4 (0.37) CHRM2CHRM1RRM1RRM2BALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102576-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed