SCHEMBL22013820

SCHEMBL22013820

COC(=O)c1cnc2c(c1)c(I)nn2COCC[Si](C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
DGAT1 O75907 8/20 0.36
MAPT P10636 1/20 0.33
KLKB1 P03952 1/20 0.32
ATM Q13315 1/20 0.32
MAPK1 P28482 1/20 0.32
ABHD6 Q9BV23 1/20 0.31
FAAH O00519 1/20 0.31
MERTK Q12866 1/20 0.31
GAA P10253 1/20 0.31
RAB9A P51151 1/20 0.31
PSMD14 O00487 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29900853 1.00 NPC1 (0.39) NPC1DGAT1MAPTKLKB1ATM
SCHEMBL30908117 0.87 NPC1 (0.37) NPC1DGAT1MAPTKLKB1ATM
SCHEMBL30908118 0.87 NPC1 (0.37) NPC1DGAT1MAPTKLKB1ATM
SCHEMBL22013944 0.87 NPC1 (0.37) NPC1DGAT1MAPTKLKB1ATM
SCHEMBL18547984 0.81 NPC1 (0.47) NPC1DGAT1MAPTKLKB1ABHD6
SCHEMBL27077167 0.81 P2RY12 (0.35) NPC1KLKB1RAB9A
SCHEMBL29900915 0.79 DGAT1 (0.38) NPC1DGAT1
SCHEMBL1593371 0.79 DGAT1 (0.38) NPC1DGAT1
SCHEMBL19250755 0.79 NPC1 (0.32) NPC1DGAT1MAPT
SCHEMBL27215111 0.79 DGAT1 (0.38) NPC1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098720-A1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed