SCHEMBL22015634

SCHEMBL22015634

c1cc(-n2cnnc2)co1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
QPCT Q16769 1/20 0.34
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28541808 0.75 MAPT (0.40) CYP1A2
SCHEMBL21241321 0.71 CYP2E1 (0.49) CYP1A2CYP2C9MAOAMAOB
SCHEMBL9594869 0.68 KMT2A (0.41)
SCHEMBL22952501 0.68
SCHEMBL7863204 0.67 CHKA (0.43)
SCHEMBL28170375 0.67
SCHEMBL16040168 0.67 NPC1 (0.58) CYP1A2MAOAMAOB
SCHEMBL25589622 0.66 NOTUM (0.50) CYP1A2CYP2C9MAOA
SCHEMBL4869797 0.65 ALDH1A1 (0.43) CYP1A2
SCHEMBL4138501 0.62 ALDH1A1 (0.31) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3218372-B1 MORPHOLINE AND 1,4-OXAZEPANE AMIDES AS SOMATOSTATIN RECEPTOR SUBTYPE 4 (SSTR4) AGONISTS BOEHRINGER INGELHEIM INT (DE) 2020-05-20 EP disclosed