SCHEMBL22019128

SCHEMBL22019128

COC1CCN(c2ncc(C(=O)c3cccc(C(F)(F)F)c3)s2)C1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCD O00767 4/20 0.52
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
RAF1 P04049 1/20 0.42
BRAF P15056 1/20 0.42
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
VNN1 O95497 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
PCSK9 Q8NBP7 1/20 0.41
MLYCD O95822 4/20 0.40
LIPG Q9Y5X9 1/20 0.40
PIM1 P11309 1/20 0.40
ACACB O00763 1/20 0.40
TMPRSS15 P98073 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22019150 0.94 SCD (0.47) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962769 0.94 SCD (0.47) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962751 0.92 SCD (0.44) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL22019127 0.86 RAF1 (0.42) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962431 0.86 RAF1 (0.42) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962446 0.86 SCD (0.46) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962542 0.85 RAF1 (0.48) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962674 0.84 SCD (0.47) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL21962458 0.83 SCD (0.46) SCDCYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL22020545 0.83 HDAC3 (0.44) SCDCYP2C9CYP2C19KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed