SCHEMBL2203102

SCHEMBL2203102

Cc1nn(-c2cccc(OC(F)(F)F)c2)c(C)c1C(=O)N1CCC(N(C)C2CCOCC2)C1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
MCHR1 Q99705 2/20 0.41
CHRM4 P08173 3/20 0.41
OPRM1 P35372 1/20 0.40
CACNA2D1 P54289 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
NOTUM Q6P988 1/20 0.38
SCN9A Q15858 2/20 0.38
PIM1 P11309 3/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
NPY5R Q15761 1/20 0.38
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CACNA1B Q00975 1/20 0.37
GPR119 Q8TDV5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2203098 1.00 KMT2A (0.45) KMT2AMCHR1CHRM4OPRM1CACNA2D1
SCHEMBL2202933 0.89 MCHR1 (0.47) KMT2AMCHR1NPSR1
SCHEMBL2202927 0.89 MCHR1 (0.47) KMT2AMCHR1NPSR1
SCHEMBL13973770 0.87 KMT2A (0.42) KMT2AMCHR1OPRM1CACNA2D1MAPT
SCHEMBL2197635 0.85 KMT2A (0.53) KMT2AOPRM1CACNA2D1NOTUMSCN9A
SCHEMBL2200002 0.85 KMT2A (0.47) KMT2AOPRM1CACNA2D1NOTUMSCN9A
SCHEMBL2203346 0.85 KMT2A (0.45) KMT2ANOTUMSCN9APIM1SCN10A
SCHEMBL2201648 0.83 KMT2A (0.49) KMT2APIM1NPY5RMAPTRAB9A
SCHEMBL2199925 0.82 KMT2A (0.50) KMT2AMCHR1SCN9ASCN10AMAPT
SCHEMBL27788063 0.81 KMT2A (0.49) KMT2AOPRM1CACNA2D1NOTUMSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977358-B2 Pyrazol derivatives HOFFMANN-LA ROCHE INC. (US) 2011-07-12 US disclosed