SCHEMBL22034178

SCHEMBL22034178

COc1ccc(C(OC[C@H]2O[C@@H](n3cnc4c(=O)[nH]c(NC(=O)C(C)C)nc43)[C@@H](O[PH](=O)Oc3ccccc3)[C@@H]2O[Si](C)(C)C(C)(C)C)(c2ccccc2)c2ccc(OC)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYMP P19971 12/20 0.47
KDM4E B2RXH2 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
NT5E P21589 1/20 0.36
HPGD P15428 1/20 0.35
ADORA1 P30542 2/20 0.33
HINT1 P49773 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20481728 0.96 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL19493439 0.95 TYMP (0.48) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL21305111 0.94 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL18490335 0.94 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL17304193 0.94 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL22034286 0.94 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL19493361 0.93 TYMP (0.48) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL25436741 0.93 TYMP (0.53) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL18992250 0.91 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E
SCHEMBL17304194 0.91 TYMP (0.49) TYMPKDM4ETAS1R3TAS1R1NT5E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3891164-A1 CYCLIC DI-NUCLEOTIDE COMPOUNDS AS STING AGONISTS Merck Sharp & Dohme Corp. (US) 2021-10-13 EP disclosed
WO-2020117625-A1 CYCLIC DI-NUCLEOTIDE COMPOUNDS AS STING AGONISTS MERCK SHARP & DOHME CORP. (US) 2020-06-11 WO disclosed