SCHEMBL22034758

SCHEMBL22034758

C[C@@H]1CNCCN1c1nc(Nc2cc(C(C)(C)C)[nH]n2)c2cc[nH]c2n1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SPAST Q9UBP0 2/20 0.74
IGF1R P08069 5/20 0.43
ROCK2 O75116 4/20 0.40
ROCK1 Q13464 3/20 0.39
PAK4 O96013 6/20 0.39
PAK1 Q13153 3/20 0.39
PLK4 O00444 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22034761 1.00 SPAST (0.74) SPASTIGF1RROCK2ROCK1PAK4
SCHEMBL22035049 0.85 SPAST (1.00) SPASTIGF1RPAK4PAK1
SCHEMBL22035048 0.85 SPAST (1.00) SPASTIGF1RPAK4PAK1
SCHEMBL22072741 0.83 SPAST (0.76) SPASTIGF1RROCK2ROCK1PAK4
SCHEMBL22072528 0.82 SPAST (0.75) SPASTIGF1RROCK2ROCK1PAK4
SCHEMBL22072737 0.82 SPAST (0.75) SPASTIGF1RROCK2ROCK1PAK4
SCHEMBL22072740 0.81 SPAST (0.76) SPASTIGF1RROCK2ROCK1PAK4
SCHEMBL22072742 0.81 SPAST (0.72) SPASTIGF1RROCK2ROCK1PAK4
SCHEMBL2044426 0.78 SPAST (0.51) SPASTROCK2ROCK1PAK4
SCHEMBL22035098 0.76 SPAST (1.00) SPASTIGF1RROCK2ROCK1PAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020118183-A1 2,4-DIAMINOPYRIMIDINE BICYCLES FOR TREATING CANCER KAPOOR TARUN M (US) 2020-06-11 WO disclosed