SCHEMBL22041432

SCHEMBL22041432

CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCC(CCO[N+](=O)[O-])CC4)ccc3OCC)nc12

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.75
HDAC1 Q13547 1/20 0.75
HDAC2 Q92769 1/20 0.75
HDAC6 Q9UBN7 1/20 0.75
PDE3B Q13370 4/20 0.74
PDE3A Q14432 4/20 0.74
PDE2A O00408 1/20 0.74
ABCC4 O15439 1/20 0.74
ABCC5 O15440 1/20 0.74
PDE6D O43924 1/20 0.74
PDE8A O60658 1/20 0.74
PDE9A O76083 1/20 0.74
ABCB11 O95342 1/20 0.74
CYP3A4 P08684 1/20 0.74
HTR1A P08908 1/20 0.74
PDE6A P16499 1/20 0.74
PDE6G P18545 1/20 0.74
PDE4A P27815 1/20 0.74
ADORA2A P29274 1/20 0.74
ADORA1 P30542 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22043079 0.96 PDE5A (0.74) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL23370711 0.94 PDE5A (0.70) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL24239380 0.91 PDE5A (0.71) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL21995695 0.91 PDE5A (0.71) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL31064951 0.91 PDE5A (0.71) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL24239278 0.91 PDE5A (0.71) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL22041040 0.90 PDE5A (0.84) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL24239354 0.90 PDE5A (0.70) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL21995286 0.90 PDE5A (0.72) PDE5AHDAC1HDAC2HDAC6PDE3B
SCHEMBL29440268 0.90 PDE5A (0.72) PDE5AHDAC1HDAC2HDAC6PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020109354-A1 NOVEL DUAL MODE OF ACTION SOLUBLE GUANYLATE CYCLASE ACTIVATORS AND PHOSPHODIESTERASE INHIBITORS AND USES THEREOF TOPADUR PHARMA AG (CH) 2020-06-04 WO disclosed