SCHEMBL220487

SCHEMBL220487

NC(=O)c1ccncn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29564726 1.00
SCHEMBL27599895 0.98
Hydrochloric Acid SCHEMBL30986896 0.98 P2RX7 (0.60)
Hydrochloric Acid SCHEMBL27472830 0.98 P2RX7 (0.60)
SCHEMBL29495233 0.98 P2RX7 (0.60)
Hydrochloric Acid SCHEMBL25429260 0.98 P2RX7 (0.60)
Benzene SCHEMBL14741825 0.96 P2RX7 (0.58)
Trimethylammonium SCHEMBL27900614 0.92 P2RX7 (0.55)
Succinic Acid SCHEMBL4542376 0.89 P2RX7 (0.56)
Trifluoroacetic Acid SCHEMBL30547497 0.87 P2RX7 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1132 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250230154-A1 COMPOUND HAVING SHP2 PROTEIN DEGRADING ACTIVITY, AND MEDICAL USES THEREOF UBIX THERAPEUTICS, INC. (KR) 2025-07-17 US claimed
CN-120092003-A CDK protein degrading agents, pharmaceutical compositions and therapeutic uses 拜欧斯瑞克斯公司 2025-06-03 CN claimed
EP-3728234-B1 RADIOLABELED COMPOUNDS HOFFMANN LA ROCHE (CH) 2025-05-14 EP claimed
CN-119907790-A Pyrazole amide insecticidal agents FMC公司 2025-04-29 CN claimed
EP-3827831-B1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NONALCOHOLIC STEATOHEPATITIS J2H BIOTECH INC (KR) 2025-03-26 EP claimed
EP-4522613-A1 CDK PROTEIN DEGRADERS, PHARMACEUTICAL COMPOSITIONS, AND THERAPEUTIC APPLICATIONS Biotheryx, Inc. (US) 2025-03-19 EP claimed
CN-119504710-A PROTACs compound for targeted degradation of PRMT5 and application thereof 昆明医科大学 2025-02-25 CN claimed
EP-4069691-B1 SUBSTITUTED TETRAHYDROFURANS AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMA (US) 2024-09-18 EP claimed
CN-118530286-A Double-function pyrimidine monoamide ligand-based complex with efficient heterogeneous organic catalysis and electrocatalytic function and application thereof 渤海大学 2024-08-23 CN claimed
US-12011443-B2 Pharmaceutical composition for preventing or treating nonalcoholic steatohepatitis J2H BIOTECH INC. (KR) 2024-06-18 US claimed
WO-2004019933-A1 METHOD OF PREVENTING OR TREATING ATHEROSCLEROSIS OR RESTENOSIS PHARMACIA & UPJOHN COMPANY (US) 2004-03-11 WO claimed
CN-1407985-A Heterocyclic dihydropyrimidines as potassium channel inhibitors BRISTOL MYERS SQUIBB CO (US) 2003-04-02 CN claimed
WO-2002048116-A2 INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-06-20 WO claimed
CN-1332743-A Cell adhesion-inhibiting antinflammatory compounds ABBOTT CO (US) 2002-01-23 CN claimed
EP-0522915-B1 Pyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics SYNTHELABO (FR) 1996-03-13 EP claimed
US-5330985-A Adrenergic blocking agents; urogenital disorders SYNTHELABO (FR) 1994-07-19 US claimed
US-5244901-A Multistage preparation by starting with a phenylpiperazine and an epoxide or chloro alcohol containing a phthalimido group; use to treat disorders involving hyperactivity of the alpha 1-adrenergic system SYNTHELABO (FR) 1993-09-14 US claimed
EP-0522915-A1 Pyrimidine-4-carboxamide derivatives, their preparation and their use in therapeutics SYNTHELABO (FR) 1993-01-13 EP claimed
CN-1067884-A Pyrimidine-4-carboxamides derivatives and method for making and medical applications SYNTHELABO (FR) 1993-01-13 CN claimed
EP-0022494-B1 BETA-LACTAM-COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC AGENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1983-02-23 EP claimed