SCHEMBL22048740

SCHEMBL22048740

CNC(=O)/C(N)=C/N(N)Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
AOC3 Q16853 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
LMNA P02545 1/20 0.38
ALDH1A1 P00352 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PLA2G10 O15496 1/20 0.37
PLA2G2A P14555 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19980450 0.84 AOC3 (0.44) NPC1RAB9AAOC3SMN1; SMN2CA12
SCHEMBL22737287 0.82 AOC3 (0.42) NPC1RAB9AAOC3SMN1; SMN2CA12
SCHEMBL23189283 0.79 AOC3 (0.44) NPC1RAB9AAOC3SMN1; SMN2KMT2A
SCHEMBL24310595 0.78 CES2 (0.42) NPC1RAB9AAOC3SMN1; SMN2KMT2A
SCHEMBL19216110 0.77 AOC3 (0.52) NPC1RAB9AAOC3SMN1; SMN2CA12
SCHEMBL20344592 0.76 TDP1 (0.39) NPC1RAB9AAOC3CA12CA9
SCHEMBL23189268 0.75 HPGD (0.41) NPC1RAB9AAOC3KMT2AMEN1
SCHEMBL19654872 0.75 AOC3 (0.48) NPC1RAB9AAOC3CA12CA9
SCHEMBL23011657 0.73
SCHEMBL23337476 0.72 AOC3 (0.42) NPC1RAB9AAOC3SMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3375780-B1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2020-06-03 EP disclosed