SCHEMBL22054063

SCHEMBL22054063

CCOC(=O)c1c2c(n(CC(=O)OC(C)(C)C)c1CC)CC1C(C)C21

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.33
IGF1R P08069 1/20 0.33
GAA P10253 3/20 0.32
ALDH1A1 P00352 4/20 0.31
HPGD P15428 3/20 0.31
KDM4E B2RXH2 3/20 0.31
HSD17B10 Q99714 2/20 0.31
MAPT P10636 2/20 0.31
TSHR P16473 2/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
KMT2A Q03164 1/20 0.30
POLB P06746 1/20 0.30
CASP1 P29466 1/20 0.30
KLK7 P49862 1/20 0.30
CASP7 P55210 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
GPR119 Q8TDV5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21764828 0.83 IGF1R (0.34) ADORA1IGF1RGAAALDH1A1HPGD
SCHEMBL21764830 0.76 ALDH1A1 (0.47) ADORA1IGF1RGAAALDH1A1HPGD
SCHEMBL23959588 0.75 STAT3 (0.33) ADORA1ALDH1A1TSHRKMT2ASMN1; SMN2
SCHEMBL23959619 0.75 STAT3 (0.33) ADORA1ALDH1A1TSHRKMT2ASMN1; SMN2
SCHEMBL21939479 0.65 CNR2 (0.34) ALDH1A1HPGDMAPTKMT2ASMN1; SMN2
SCHEMBL23959581 0.63 ALDH1A1 (0.36) GAAALDH1A1HPGDKDM4EHSD17B10
SCHEMBL24878671 0.61 IDO1 (0.36) ALDH1A1KDM4ETSHRKMT2ASMN1; SMN2
SCHEMBL24878539 0.61 IDO1 (0.36) ALDH1A1KDM4ETSHRKMT2ASMN1; SMN2
SCHEMBL16006626 0.60 GLA (0.31) GPR119
SCHEMBL7429634 0.59 MEN1 (0.67) ALDH1A1KDM4EHSD17B10TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020112581-A1 NOVEL SUBSTITUTED PIPERAZINE AMIDE COMPOUNDS AS INDOLEAMINE 2, 3-DIOXYGENASE (IDO) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2020-06-04 WO disclosed