SCHEMBL22065296

SCHEMBL22065296

CNc1cc(NC(=O)Nc2cccc(C(F)(F)F)c2)ccc1C

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
MAPT P10636 1/20 0.63
HTT P42858 1/20 0.63
RAB9A P51151 1/20 0.63
IDH1 O75874 12/20 0.61
ALDH1A1 P00352 1/20 0.58
GRIK1 P39086 1/20 0.58
RAF1 P04049 1/20 0.58
KDR P35968 1/20 0.57
LMNA P02545 1/20 0.57
MAPK1 P28482 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29470036 0.92 KMT2A (0.67) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL22065300 0.88 MEN1 (0.62) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL22025448 0.87 IDH1 (0.61) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL22024988 0.87 MAPT (0.62) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL22025522 0.86 MAPT (0.60) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL22025430 0.86 MEN1 (0.59) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL17131157 0.85 MAPK14 (0.72) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL19073209 0.85 BRAF (0.73) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL17079632 0.84 DDX3X (0.73) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL6371123 0.83 TRPV1 (0.67) MEN1KMT2AMAPTHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed