SCHEMBL22072049

SCHEMBL22072049

Oc1cccc(Nc2nc(Nc3cc(C4CC4)[nH]n3)c3ccccc3n2)c1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 4/20 0.72
PDK1 Q15118 1/20 0.63
ULK2 Q8IYT8 1/20 0.63
NTRK1 P04629 2/20 0.62
NTRK3 Q16288 1/20 0.58
NTRK2 Q16620 1/20 0.58
SRC P12931 4/20 0.56
GSK3B P49841 4/20 0.56
AURKA O14965 1/20 0.56
IGF1R P08069 2/20 0.56
PAK4 O96013 1/20 0.56
PAK1 Q13153 1/20 0.56
CCNA2 P20248 2/20 0.55
CDK2 P24941 2/20 0.55
TAAR1 Q96RJ0 1/20 0.53
AURKB Q96GD4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12430667 0.91 ULK1 (0.86) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL31471779 0.91 ULK1 (0.86) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL12430703 0.89 ULK1 (0.73) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL12430668 0.88 ULK1 (0.72) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL12430693 0.87 ULK1 (0.68) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL7108312 0.85 ULK1 (0.68) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL12430694 0.85 ULK1 (0.68) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL12430692 0.84 ULK1 (0.64) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL12430682 0.84 ULK1 (0.75) ULK1PDK1ULK2NTRK1NTRK3
SCHEMBL31471772 0.84 ULK1 (0.81) ULK1PDK1ULK2NTRK1NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020118183-A1 2,4-DIAMINOPYRIMIDINE BICYCLES FOR TREATING CANCER KAPOOR TARUN M (US) 2020-06-11 WO disclosed