SCHEMBL22072083

SCHEMBL22072083

CN1CC2CC(C1)N2c1nc(Nc2cc(C(C)(C)C)[nH]n2)c2ccccc2n1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SPAST Q9UBP0 2/20 0.61
PAK4 O96013 1/20 0.47
PAK1 Q13153 1/20 0.47
AURKA O14965 6/20 0.42
SRC P12931 4/20 0.42
GSK3B P49841 4/20 0.42
IGF1R P08069 4/20 0.42
ROCK2 O75116 1/20 0.41
AURKB Q96GD4 4/20 0.41
EIF2AK2 P19525 1/20 0.41
GSK3A P49840 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
ULK1 O75385 1/20 0.39
HTR3A P46098 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22035049 0.76 SPAST (1.00) SPASTPAK4PAK1IGF1R
SCHEMBL22035048 0.76 SPAST (1.00) SPASTPAK4PAK1IGF1R
SCHEMBL4073913 0.74 SPAST (0.58) SPASTAURKASRCGSK3BIGF1R
SCHEMBL7028703 0.74 AURKA (0.72) SPASTAURKASRCGSK3BAURKB
SCHEMBL22072048 0.73 SPAST (0.77) SPASTPAK4PAK1AURKAIGF1R
SCHEMBL5255520 0.68 HRH4 (0.65) PAK4PAK1AURKASRCGSK3B
SCHEMBL801474 0.68 CYP1A2 (0.63) SPASTAURKASRCGSK3BAURKB
SCHEMBL31471834 0.68 PAK4 (0.56) PAK4PAK1SRCGSK3BIGF1R
SCHEMBL22072524 0.67 PAK4 (0.83) PAK4PAK1IGF1RHRH4
SCHEMBL31471972 0.67 PAK4 (0.83) PAK4PAK1IGF1RHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020118183-A1 2,4-DIAMINOPYRIMIDINE BICYCLES FOR TREATING CANCER KAPOOR TARUN M (US) 2020-06-11 WO disclosed