SCHEMBL22089166

SCHEMBL22089166

O=CC[C@@H](Cc1ccc(F)cc1)c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
CNR1 P21554 2/20 0.39
NOS2 P35228 1/20 0.38
MDM2 Q00987 1/20 0.38
SLC6A4 P31645 1/20 0.38
BCL2A1 Q16548 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
CYP19A1 P11511 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
GMNN O75496 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2088573 0.92 CYP19A1 (0.40) SLC6A4POLBCYP19A1HTTSLC6A2
SCHEMBL28615059 0.84 MEN1 (0.44) PPARGPPARACNR1SLC6A4MEN1
SCHEMBL3136328 0.79 GABBR2 (0.43) RAB9AHTTSLC6A3
SCHEMBL16439493 0.77 GABBR2 (0.58) PPARGPPARATHRBMEN1KMT2A
SCHEMBL29120227 0.76 GABBR2 (0.39) SLC6A4HTTSLC6A2SLC6A3
SCHEMBL11225612 0.76 MEN1 (0.40) MAPTTHRBMEN1KMT2AHTT
SCHEMBL28819403 0.75 PPARG (0.45) PPARGPPARAMAPTTHRBCNR1
SCHEMBL18382609 0.73 GABBR2 (0.56) MAPTTHRBSLC6A4MEN1KMT2A
SCHEMBL26922771 0.73 GABBR2 (0.56) MAPTTHRBSLC6A4MEN1KMT2A
SCHEMBL26923676 0.73 GABBR2 (0.56) MAPTTHRBSLC6A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3027593-B1 PIPERAZINE DERIVATIVES AS HIV PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2020-06-10 EP disclosed