SCHEMBL2208923

SCHEMBL2208923

O=C(NCC1CCCCC1)Oc1ccc2cc(OCCCN3CCCCC3)ccc2n1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.55
AVPR1B P47901 3/20 0.51
PDE3B Q13370 3/20 0.45
PDE3A Q14432 3/20 0.45
TLR9 Q9NR96 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
MAOB P27338 1/20 0.44
SCN7A Q01118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1381004 0.85 HRH3 (0.65) HRH3AVPR1BPDE3BPDE3A
SCHEMBL2209226 0.85 HRH3 (0.51) HRH3AVPR1BPDE3BPDE3A
SCHEMBL2211945 0.82 HRH3 (0.54) HRH3AVPR1B
SCHEMBL2209034 0.81 HRH3 (0.52) HRH3PDE3BPDE3ATLR9TLR7
SCHEMBL2211880 0.80 HRH3 (0.51) HRH3AVPR1BPDE3BPDE3AMAOB
SCHEMBL4501875 0.80 HRH3 (0.63) HRH3AVPR1BMAOB
SCHEMBL2208812 0.77 HRH3 (0.54) HRH3AVPR1BMAOBSCN7A
SCHEMBL2242065 0.77 HRH3 (0.57) HRH3
SCHEMBL4490636 0.77 HRH3 (0.64) HRH3AVPR1BMAOB
SCHEMBL2212122 0.76 HRH3 (0.51) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805166-B1 QUINOLINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-07-27 EP claimed