SCHEMBL22100726

SCHEMBL22100726

CNC(=O)c1cc(CBr)cc(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.50
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50
GAA P10253 4/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 3/20 0.45
HPGD P15428 1/20 0.45
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44
TUBB2A Q13885 1/20 0.44
TUBB8 Q3ZCM7 1/20 0.44
TUBA3E Q6PEY2 1/20 0.44
TUBA1A Q71U36 1/20 0.44
TUBA1C Q9BQE3 1/20 0.44
TUBB6 Q9BUF5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3930458 0.85 PLK1 (0.51) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL3930459 0.85 PLK1 (0.51) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL3937664 0.84 PLK1 (0.50) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL20145771 0.84 PLK1 (0.50) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL29581270 0.83 CA1 (0.47) GAAKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL1096840 0.83 CA1 (0.47) GAAKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL14288600 0.83 PLK1 (0.54) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL7959771 0.82 PLK1 (0.64) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL89288 0.82 NPC1 (0.56) GAAKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL5270681 0.81 CA1 (0.47) KDM4ELMNASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321261-B1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES CURIS INC (US) 2020-06-17 EP disclosed