SCHEMBL20145771

SCHEMBL20145771

BCc1cc(OC)cc(C(=O)NC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.50
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50
GAA P10253 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX12 P18054 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HPGD P15428 1/20 0.42
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3930459 0.85 PLK1 (0.51) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL3930458 0.85 PLK1 (0.51) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL22100726 0.84 PLK1 (0.50) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL3937664 0.84 PLK1 (0.50) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL14288600 0.83 PLK1 (0.54) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL7959771 0.82 PLK1 (0.64) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL1911352 0.82 NPC1 (0.56) GAAKDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL3940442 0.80 GAA (0.51) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL17414596 0.78 PLK1 (0.55) PLK1HSD17B1HSD17B2GAAKDM4E
SCHEMBL12430522 0.76 PLK1 (0.56) PLK1HSD17B1HSD17B2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321261-A1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES Curis, Inc. (US) 2018-05-16 EP disclosed