SCHEMBL22102488

SCHEMBL22102488

Cc1ccc(C(=O)Cc2ccc3ncc(Br)cc3c2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
GRM1 Q13255 1/20 0.39
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
KCNE1 P15382 2/20 0.38
KCNQ1 P51787 2/20 0.38
KCNQ5 Q9NR82 1/20 0.38
MAPT P10636 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MGLL Q99685 1/20 0.35
PKM P14618 1/20 0.35
MAOB P27338 1/20 0.34
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.34
PTGFR P43088 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22075469 0.90 VNN1 (0.38) GRM1KCNQ3KCNQ2KCNQ5MAOB
SCHEMBL22103180 0.81 PIK3CA (0.40) HDAC1HDAC6MAPTALDH1A1
SCHEMBL26003352 0.79 KDM4E (0.42) HDAC6GRM1MAPTSMN1; SMN2ALDH1A1
SCHEMBL22075266 0.77 ERCC5 (0.40) HDAC1HDAC6GRM1KCNQ3KCNQ2
SCHEMBL22075124 0.76 PIK3CA (0.40) SMN1; SMN2LMNA
SCHEMBL22074806 0.75 PIK3CA (0.42) HDAC1HDAC6MAPTLMNATP53
SCHEMBL3158828 0.75 GAA (0.44) MAPTALDH1A1LMNAHPGD
SCHEMBL23389840 0.74 NPC1 (0.40) HDAC1HDAC6GRM1SMN1; SMN2LMNA
SCHEMBL29796631 0.74 NPC1 (0.40) HDAC1HDAC6GRM1SMN1; SMN2LMNA
SCHEMBL29151068 0.73 MAOB (0.50) MAPTSMN1; SMN2ALDH1A1HPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020123453-A2 ALK5 INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC (US) 2020-06-18 WO disclosed