SCHEMBL22111140

SCHEMBL22111140

N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.53
GSTK1 Q9Y2Q3 1/20 0.53
GLO1 Q04760 1/20 0.53
FOLH1 Q04609 7/20 0.49
RIMKLA Q8IXN7 1/20 0.49
NAALAD2 Q9Y3Q0 1/20 0.49
NOD1 Q9Y239 2/20 0.46
GRM8 O00222 1/20 0.44
GRM6 O15303 1/20 0.44
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
GSR P00390 1/20 0.44
CYP1A2 P05177 1/20 0.44
GRIK1 P39086 1/20 0.44
GRM5 P41594 1/20 0.44
GRIA1 P42261 1/20 0.44
GRIA2 P42262 1/20 0.44
GRIA3 P42263 1/20 0.44
SLC1A3 P43003 1/20 0.44
SLC1A2 P43004 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29695437 0.97 PTGS1 (0.51) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL30099681 0.97 PTGS1 (0.51) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL30292792 0.97 PTGS1 (0.52) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL29695622 0.96 GLO1 (0.49) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL30099464 0.94 PTGS1 (0.51) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL30099536 0.94 PTGS1 (0.51) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL30099480 0.94 PTGS1 (0.51) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL29742960 0.94 PTGS1 (0.51) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL30099519 0.93 GLO1 (0.48) PTGS1GSTK1GLO1FOLH1RIMKLA
SCHEMBL29526001 0.93 PTGS1 (0.50) PTGS1GSTK1GLO1FOLH1RIMKLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666788-A1 HEMIASTERLIN DERIVATIVES AND ANTIBODY-DRUG CONJUGATES INCLUDING SAME Sumitomo Dainippon Pharma Co., Ltd. (JP) 2020-06-17 EP disclosed