SCHEMBL2212145

SCHEMBL2212145

CC(C)(C)OC(=O)Nc1cccc(Nc2nc(-c3cccc4c3oc3ccccc34)cc3ccnn23)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.39
TDP2 O95551 1/20 0.37
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
SYK P43405 1/20 0.37
RORC P51449 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
ACSS2 Q9NR19 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35
CCKBR P32239 1/20 0.34
F2RL3 Q96RI0 1/20 0.34
CYP17A1 P05093 1/20 0.34
IDO1 P14902 1/20 0.33
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33
MAPT P10636 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2215145 0.94 BRD4 (0.36) BRD4TDP2TOP2ATOP2BTLR7
SCHEMBL2214770 0.89 NAMPT (0.34) BRD4F2RL3MAPT
SCHEMBL2214311 0.86 KCNK9 (0.44) SYKCA1MAPT
SCHEMBL2215562 0.85 SUV39H2 (0.34) BRD4CCKBR
SCHEMBL2215249 0.84 SMN1; SMN2 (0.37) MAPT
SCHEMBL2213364 0.83 NAMPT (0.36) BRD4CCKBRMAPT
SCHEMBL2214124 0.82 MAPT (0.49) MAPT
SCHEMBL2214698 0.82 BRD4 (0.38) BRD4CCKBRMAPT
SCHEMBL2214495 0.82 P2RY14 (0.47) MAPT
SCHEMBL2214767 0.82 SMN1; SMN2 (0.38) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797096-B1 PYRAZOLOPYRIMIDINES AS INHIBITORS OF PROTEIN KINASE B (AKT) BAYER SCHERING PHARMA AG (DE) 2011-07-27 EP disclosed