SCHEMBL2212947

SCHEMBL2212947

CCCN(c1ccccc1C(N)=O)S(C)(=O)=O

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.44
ESR1 P03372 7/20 0.41
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 2/20 0.39
NR1I2 O75469 1/20 0.39
LMNA P02545 1/20 0.39
CHRM2 P08172 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADRA2A P08913 1/20 0.39
MAPT P10636 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HSD17B10 Q99714 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10613988 0.78 TP53 (0.49) TP53KMT2AALDH1A1MEN1NR1I2
SCHEMBL28002534 0.76 KMT2A (0.66) KMT2AALDH1A1L3MBTL1MEN1MAPT
SCHEMBL7437271 0.75 TP53 (0.46) TP53KMT2AALDH1A1L3MBTL1MEN1
Hydrochloric Acid SCHEMBL30004917 0.74 KMT2A (0.64) KMT2AALDH1A1L3MBTL1MEN1MAPT
Hydrochloric Acid SCHEMBL30006002 0.74 KMT2A (0.64) KMT2AALDH1A1L3MBTL1MEN1MAPT
SCHEMBL1290816 0.74 ESR1 (0.62) ESR1KMT2AALDH1A1MEN1CYP3A4
SCHEMBL11830362 0.74 KMT2A (0.46) TP53ESR1KMT2AALDH1A1
SCHEMBL7554537 0.73 KMT2A (0.54) ESR1KMT2AALDH1A1L3MBTL1LMNA
SCHEMBL6417177 0.73 KMT2A (0.43) TP53KMT2AALDH1A1L3MBTL1MEN1
SCHEMBL10639178 0.72 KMT2A (0.54) TP53ESR1KMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689713-B1 BENZYLETHER AND BENZYLAMINO BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER S DISEASE MERCK SHARP & DOHME (US) 2011-07-27 EP disclosed