SCHEMBL2213775

SCHEMBL2213775

CCS(=O)(=O)Nc1cc(C(=O)OC)cc(N(Cc2ccccc2)C[C@@H]2C[C@H]2C)n1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.42
NR3C1 P04150 3/20 0.39
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5155015 0.92 BACE1 (0.41) BACE1NR3C1HPGD
SCHEMBL4512858 0.83 BACE1 (0.55) BACE1NR3C1KDM4EALDH1A1
SCHEMBL2020790 0.73 BACE1 (0.52) BACE1
SCHEMBL12578837 0.72 BACE1 (0.59) BACE1
SCHEMBL2027404 0.71 BACE1 (0.59) BACE1
SCHEMBL2027128 0.71 BACE1 (0.59) BACE1
SCHEMBL8264847 0.69 BACE1 (0.39) BACE1
SCHEMBL5653669 0.69 BACE1 (0.54) BACE1ALDH1A1
SCHEMBL5653668 0.69 BACE1 (0.54) BACE1ALDH1A1
SCHEMBL4740207 0.67 BACE1 (0.38) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689713-B1 BENZYLETHER AND BENZYLAMINO BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER S DISEASE MERCK SHARP & DOHME (US) 2011-07-27 EP disclosed