SCHEMBL22143602

SCHEMBL22143602

COC(=O)C(Cc1cc(OS(=O)(=O)C(F)(F)F)ccc1Cl)NC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.43
SCN9A Q15858 3/20 0.40
BCL2 P10415 5/20 0.40
CYP3A4 P08684 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
MCL1 Q07820 1/20 0.40
CTSS P25774 2/20 0.40
CTSK P43235 2/20 0.40
PTPN1 P18031 1/20 0.39
MMP13 P45452 1/20 0.39
CTSL P07711 1/20 0.39
TACR1 P25103 2/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
ABCB1 P08183 1/20 0.37
ACE P12821 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22143911 1.00 KLK5 (0.43) KLK5SCN9ABCL2CYP3A4SCN10A
SCHEMBL2890943 0.87 CTSS (0.47) KLK5SCN9ABCL2CTSSCTSK
SCHEMBL864694 0.83 KLK5 (0.53) KLK5BCL2CTSSCTSKPTPN1
SCHEMBL1819934 0.83 KLK5 (0.53) KLK5BCL2CTSSCTSKPTPN1
SCHEMBL7442384 0.83 KLK5 (0.53) KLK5BCL2CTSSCTSKPTPN1
SCHEMBL31277258 0.82 MAPT (0.49) KLK5SCN9ACYP3A4SCN10ACTSS
SCHEMBL22425268 0.81 KLK5 (0.47) KLK5SCN9ACYP3A4SCN10ACTSS
SCHEMBL28599848 0.81 KLK5 (0.47) KLK5SCN9ACYP3A4SCN10ACTSS
SCHEMBL27564123 0.81 TACR1 (0.50) KLK5SCN9ACYP3A4SCN10ACTSS
SCHEMBL31689558 0.80 KLK5 (0.48) KLK5SCN9ACYP3A4SCN10ACTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164448-A Amino acid anilines as small molecule modulators of IL-17 利奥制药有限公司 2021-07-23 CN disclosed
WO-2020127685-A1 AMINO-ACID ANILIDES AS SMALL MOLECULE MODULATORS OF IL-17 LEO PHARMA A/S (DK) 2020-06-25 WO disclosed