SCHEMBL22146341

SCHEMBL22146341

O=C(NC1CC2CCC(C1)N2)c1ccc2c(c1)OCCO2

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.67
RAB9A P51151 7/20 0.67
CHRNA7 P36544 2/20 0.60
MAPK11 Q15759 1/20 0.57
MAPK14 Q16539 1/20 0.57
NFKB1 P19838 2/20 0.56
NFKB2 Q00653 2/20 0.56
RELA Q04206 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
TP53 P04637 1/20 0.56
HPGD P15428 1/20 0.56
KMT2A Q03164 1/20 0.54
CYP2C9 P11712 1/20 0.51
ACHE P22303 1/20 0.49
SMYD3 Q9H7B4 1/20 0.49
KDM4E B2RXH2 1/20 0.49
MAPK1 P28482 1/20 0.49
PKM P14618 1/20 0.49
MAOB P27338 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2797986 0.81 NPC1 (0.75) NPC1RAB9ACHRNA7MAPK11MAPK14
SCHEMBL29779541 0.81 SMYD3 (0.67) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL17592010 0.81 SMYD3 (0.67) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL17592011 0.81 SMYD3 (0.67) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL3214001 0.77 NPC1 (0.72) NPC1RAB9ACHRNA7MAPK11MAPK14
SCHEMBL6820557 0.77 TAS1R3 (0.52) NPC1RAB9ACHRNA7HPGDKMT2A
SCHEMBL5232236 0.76 NPC1 (0.56) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL6291512 0.76 CHRNA7 (0.89) NPC1RAB9ACHRNA7MAPK11MAPK14
SCHEMBL6288321 0.75 CHRNA7 (1.00) NPC1RAB9ACHRNA7MAPK11MAPK14
SCHEMBL6288322 0.75 CHRNA7 (1.00) NPC1RAB9ACHRNA7MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906216-B1 INHIBITORS OF DNA GYRASE FOR THE TREATMENT OF BACTERIAL INFECTIONS KUMAR AJAY (GB) 2020-06-24 EP disclosed