SCHEMBL22147393

SCHEMBL22147393

c1ccc(-c2ccnc(-c3cnccn3)n2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
KDM4E B2RXH2 7/20 0.53
TP53 P04637 4/20 0.53
LMNA P02545 3/20 0.53
CCR1 P32246 3/20 0.53
CCR5 P51681 3/20 0.53
CCR8 P51685 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
ALOX15 P16050 3/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
TDP1 Q9NUW8 2/20 0.53
HTT P42858 2/20 0.53
ALPL P05186 1/20 0.53
HSP90AA1 P07900 1/20 0.53
ALPI P09923 1/20 0.53
ALPG P10696 1/20 0.53
MAPK1 P28482 1/20 0.53
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dipyridyl SCHEMBL28077341 0.89 KDM4E (0.58) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL20169526 0.87 NPC1 (0.44) NPC1RAB9AKDM4EHTTHSP90AA1
SCHEMBL776048 0.85 KDM4E (0.67) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL2062004 0.82 KDM4E (0.67) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL29907668 0.82 KDM4E (0.67) NPC1RAB9AKDM4ETP53LMNA
Dipyridyl SCHEMBL6050743 0.82 KDM4E (0.67) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL31140235 0.82 KDM4E (0.67) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL6535045 0.81 KDM4E (0.67) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL19944117 0.79 KDM4E (0.59) NPC1RAB9AKDM4ETP53LMNA
SCHEMBL27946179 0.79 KDM4E (0.59) NPC1RAB9AKDM4ETP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3670509-A1 INHIBITORS OF INV(16) LEUKEMIA The University of Virginia Patent Foundation (US) 2020-06-24 EP disclosed