SCHEMBL221526

SCHEMBL221526

C=C(Cl)C([NH])=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL690502 0.73
SCHEMBL991031 0.71
SCHEMBL144716 0.70
SCHEMBL28875041 0.70 LDHA (0.33)
SCHEMBL66157 0.70
SCHEMBL2864068 0.70
SCHEMBL338357 0.70
SCHEMBL7513194 0.70
SCHEMBL65175 0.67
SCHEMBL35038 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 233 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3268375-B1 PHOTOCHROMIC THIENOCHROMENE COMPOUNDS TRANSITIONS OPTICAL INC (US) 2022-06-15 EP claimed
EP-3071576-B9 PHOTOCHROMIC INDENO-FUSED RING PYRAN COMPOUNDS TRANSITIONS OPTICAL INC (US) 2021-12-22 EP claimed
EP-3645540-B1 SILOLE AND GERMOLE FUSED RING PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL LTD (IE) 2021-11-03 EP claimed
EP-3071576-B1 PHOTOCHROMIC INDENO-FUSED RING PYRAN COMPOUNDS TRANSITIONS OPTICAL INC (US) 2021-08-18 EP claimed
CN-105199708-B Photochromic compounds 光学转变公司 2020-10-27 CN claimed
US-20200172798-A1 Silole and Germole Fused Ring Photochromic Compounds TRANSITIONS OPTICAL, LTD. (IE) 2020-06-04 US claimed
EP-3645540-A1 SILOLE AND GERMOLE FUSED RING PHOTOCHROMIC COMPOUNDS Transitions Optical, Ltd. (IE) 2020-05-06 EP claimed
EP-3621958-A1 PHOTOCHROMIC INDENO FUSED PHENANTHRENOPYRAN COMPOUNDS Transitions Optical, Ltd. (IE) 2020-03-18 EP claimed
US-20200048216-A1 Photochromic Indeno Fused Phenanthrenopyran Compounds TRANSITIONS OPTICAL, LTD. (IE) 2020-02-13 US claimed
EP-2370420-B9 PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL INC (US) 2019-11-13 EP claimed
WO-2010065406-A1 ALIGNMENT FACILITIES FOR OPTICAL DYES TRANSITIONS OPTICAL, INC. (US) 2010-06-10 WO claimed
WO-2010065393-A1 PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL, INC. (US) 2010-06-10 WO claimed
US-20090309076-A1 PHOTOCHROMIC COMPOUNDS TRANSITIONS OPTICAL, INC. (US) 2009-12-17 US claimed
US-20090146104-A1 ALIGNMENT FACILITIES FOR OPTICAL DYES TRANSITIONS OPTICAL, INC. (US) 2009-06-11 US claimed
US-20090135462-A1 CLEAR TO CIRCULAR POLARIZING PHOTOCHROMIC DEVICES AND METHODS OF MAKING THE SAME TRANSITIONS OPTICAL, INC. (US) 2009-05-28 US claimed
US-6552175-B2 1-hydroxy-2-((sulfophenyl)azo),3,(5 or 6)-disulfo-8-((4-((susbstituted aryl)amino),6-halo-s-triazin-2-yl)-naphthalene dye of given formula CIBA SPECIALTY CHEMICALS CORPORATION 2003-04-22 US claimed
EP-1247841-A2 Reactive dyes, process for their preparation and the use thereof Ciba SC Holding AG (CH) 2002-10-09 EP claimed
US-20020138922-A1 Reactive dyes, a process for their preparation and their use HUNTSMAN INTERNATIONAL LLC 2002-10-03 US claimed
WO-2000015896-A1 METHOD FOR DYEING FIBROUS MATERIALS CONTAINING CELLULOSE CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2000-03-23 WO claimed
EP-0642609-B1 PROCESS FOR THE FIXATION OF DYES CONTAINING AT LEAST ONE POLYMERISABLE DOUBLE BOND BY MEANS OF IONISING RADIATION CIBA GEIGY AG (CH) 1996-08-28 EP claimed