SCHEMBL2216178

SCHEMBL2216178

COc1ccccc1-c1ccc(-c2cc3ccnn3c(SC)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.43
KMT2A Q03164 2/20 0.41
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
MEN1 O00255 1/20 0.37
BLM P54132 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SQOR Q9Y6N5 1/20 0.37
PIK3R1 P27986 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2212035 0.82 SMN1; SMN2 (0.39) KMT2AMAPTKDM4EALDH1A1POLB
SCHEMBL2213882 0.82 SMN1; SMN2 (0.45) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL2211698 0.80 DHODH (0.44) DHODHKMT2AMAPTKDM4EALDH1A1
SCHEMBL2214144 0.77
SCHEMBL2213284 0.77 NPC1 (0.38) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL2214089 0.77 MAPT (0.44) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL2212151 0.76 GSK3B (0.36) DHODHKMT2AMAPTKDM4EALDH1A1
SCHEMBL2212656 0.75 SMN1; SMN2 (0.35) KMT2AMAPTKDM4EALDH1A1POLB
SCHEMBL24387355 0.74 HCRTR2 (0.34)
SCHEMBL2213701 0.72 CDK2 (0.44) KMT2AMAPTKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797096-B1 PYRAZOLOPYRIMIDINES AS INHIBITORS OF PROTEIN KINASE B (AKT) BAYER SCHERING PHARMA AG (DE) 2011-07-27 EP disclosed
EP-1797096-A2 NOVEL PYRAZOLOPYRIMIDINES Altana Pharma AG (DE) 2007-06-20 EP disclosed
WO-2006027346-A2 NOVEL PYRAZOLOPYRIMIDINES ALTANA PHARMA AG (DE) 2006-03-16 WO disclosed